Stimulation of ENaC activity by rosiglitazone is PPARγ-dependent and correlates with SGK1 expression increase.

Details

Serval ID
serval:BIB_59330169CEDE
Type
Article: article from journal or magazin.
Collection
Publications
Institution
Title
Stimulation of ENaC activity by rosiglitazone is PPARγ-dependent and correlates with SGK1 expression increase.
Journal
Journal of Membrane Biology
Author(s)
Renauld S., Tremblay K., Ait-Benichou S., Simoneau-Roy M., Garneau H., Staub O., Chraïbi A.
ISSN
1432-1424[electronic], 0022-2631[linking]
Publication state
Published
Issued date
2010
Peer-reviewed
Oui
Volume
236
Number
3
Pages
259-270
Language
english
Abstract
Thiazolidinediones (TZDs) are peroxisome proliferator-activated receptor gamma (PPARγ) agonists used to treat type 2 diabetes. TZD treatment induces side effects such as peripheral fluid retention, often leading to discontinuation of therapy. Previous studies have shown that PPARγ activation by TZD enhances the expression or function of the epithelial sodium channel (ENaC) through different mechanisms. However, the effect of TZDs on ENaC activity is not clearly understood. Here, we show that treating Xenopus laevis oocytes expressing ENaC and PPARγ with the TZD rosiglitazone (RGZ) produced a twofold increase of amiloride-sensitive sodium current (Iam), as measured by two-electrode voltage clamp. RGZ-induced ENaC activation was PPARγ-dependent since the PPARγ antagonist GW9662 blocked the activation. The RGZ-induced Iam increase was not mediated through direct serum- and glucocorticoid-regulated kinase (SGK1)-dependent phosphorylation of serine residue 594 on the human ENaC α-subunit but by the diminution of ENaC ubiquitination through the SGK1/Nedd4-2 pathway. In accordance, RGZ increased the activity of ENaC by enhancing its cell surface expression, most probably indirectly mediated through the increase of SGK1 expression.
Keywords
Animals, Cells, Cultured, Epithelial Sodium Channel/drug effects, Epithelial Sodium Channel/metabolism, Immediate-Early Proteins/metabolism, Ion Channel Gating/drug effects, Ion Channel Gating/physiology, Oocytes/drug effects, Oocytes/physiology, PPAR gamma/agonists, PPAR gamma/metabolism, Protein-Serine-Threonine Kinases/metabolism, Signal Transduction/drug effects, Signal Transduction/physiology, Statistics as Topic, Thiazolidinediones/pharmacology, Up-Regulation/drug effects, Xenopus laevis
Pubmed
Web of science
Create date
11/03/2011 13:43
Last modification date
20/10/2020 14:41
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