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Small-Molecule Protein-Protein Interaction Inhibitor of Oncogenic Rho Signaling.
10.1016/j.chembiol.2016.07.015
27593112
000384731600015
Diviani
D.
author
Raimondi
F.
author
Del Vescovo
C.D.
author
Dreyer
E.
author
Reggi
E.
author
Osman
H.
author
Ruggieri
L.
author
Gonano
C.
author
Cavin
S.
author
Box
C.L.
author
Lenoir
M.
author
Overduin
M.
author
Bellucci
L.
author
Seeber
M.
author
Fanelli
F.
author
article
2016-09-22
2016
Cell Chemical Biology
2451-9456
journal
23
9
1135-1146
A Kinase Anchor Proteins/antagonists & inhibitors
A Kinase Anchor Proteins/metabolism
Humans
Minor Histocompatibility Antigens/metabolism
Models, Molecular
Molecular Structure
Neoplasms/drug therapy
Neoplasms/metabolism
Protein Binding/drug effects
Proto-Oncogene Proteins/antagonists & inhibitors
Proto-Oncogene Proteins/metabolism
Signal Transduction/drug effects
Small Molecule Libraries/chemistry
Small Molecule Libraries/pharmacology
rho GTP-Binding Proteins/antagonists & inhibitors
rho GTP-Binding Proteins/metabolism
AKAP13 oncogene
Ras GTPases
RhoGEFs
comparative modeling
virtual screening
eng
60_published
peer-reviewed